Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water - Université de technologie de Compiègne Access content directly
Journal Articles Tetrahedron Letters Year : 2013

Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water

Abstract

A new and efficient ligandless cross-coupling reaction of 6-iodouridine with various boronic acids in the presence of Na2PdCl4 was performed at room temperature in aerobic water. The target 6-aryl analogues were obtained in moderate to good yields depending on the boronic acid nature.

Dates and versions

hal-04391353 , version 1 (12-01-2024)

Identifiers

Cite

Gérald Enderlin, Guillaume Sartori, Gwénaëlle Hervé, Christophe Len. Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water. Tetrahedron Letters, 2013, 54 (26), pp.3374-3377. ⟨10.1016/j.tetlet.2013.04.066⟩. ⟨hal-04391353⟩
4 View
0 Download

Altmetric

Share

Gmail Mastodon Facebook X LinkedIn More