Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water - Université de technologie de Compiègne Accéder directement au contenu
Article Dans Une Revue Tetrahedron Letters Année : 2013

Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water

Résumé

A new and efficient ligandless cross-coupling reaction of 6-iodouridine with various boronic acids in the presence of Na2PdCl4 was performed at room temperature in aerobic water. The target 6-aryl analogues were obtained in moderate to good yields depending on the boronic acid nature.

Domaines

Chimie

Dates et versions

hal-04391353 , version 1 (12-01-2024)

Identifiants

Citer

Gérald Enderlin, Guillaume Sartori, Gwénaëlle Hervé, Christophe Len. Synthesis of 6-aryluridines via Suzuki–Miyaura cross-coupling reaction at room temperature under aerobic ligand-free conditions in neat water. Tetrahedron Letters, 2013, 54 (26), pp.3374-3377. ⟨10.1016/j.tetlet.2013.04.066⟩. ⟨hal-04391353⟩
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